Pluripotin is a dual inhibitor of ERK1 and RasGAP with KDs of 98 nM and 212 nM, respectively. Pluripotin also inhibits RSK1, RSK2, RSK3, and RSK4 with IC50s of 0.5, 2.5, 3.3, and 10.0 µM, respectively.
Molecular Weight:
550.54
Purity:
98.86
CAS Number:
[839707-37-8]
Formula:
C27H25F3N8O2
Target:
ERK,Ribosomal S6 Kinase (RSK)
Application Notes:
Reference compound
* VAT and and shipping costs not included. Errors and price changes excepted