Lurosetron (GR-87442) is a 6-fluoro analogue of Alosetron (HY-70050A). Lurosetron is a serotonin 5-HT3 receptor antagonist. Lurosetron inhibits recombinant (rbt) CYP1A2, with an IC50 of 0.1 µM. Lurosetron also inhibits other CYP isoforms, including rbtCY
Molecular Weight:
312.34
CAS Number:
[128486-54-4]
Formula:
C17H17FN4O
Target:
5-HT Receptor
Application Notes:
Reference compound
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