TC-MCH 7c, a phenylpyridone derivative, is an orally available, selective and brain-penetrable MCH1R antagonist with an IC50 of 5.6 nM for hMCH1R[1]. TC-MCH 7c has Kis of 3.4 nM and 3.0 nM of human and mouse MCH1R, respectively[2].
Molecular Weight:
408.47
Purity:
99.79
CAS Number:
[864756-35-4]
Formula:
C24H25FN2O3
Target:
MCHR1 (GPR24)
Application Notes:
Reference compound
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