TC-E 5001 is an inhibitor of Wnt pathway that inhibits tankyrase 1/2 (TNKS1/2) via novel adenosine pocket binding, with Kds of 79 nM and 28 nM, respectively. TC-E 5001 also inhibits Axin2 and STF, with IC50s of 0.709 µM and 0.215 µM, respectively[1][2].
Molecular Weight:
409.46
CAS Number:
[865565-29-3]
Formula:
C20H19N5O3S
Target:
PARP
Application Notes:
Reference compound
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