TC-G 1005 is a potent, selective and orally active agonist of the BA receptor Takeda G protein-coupled receptor 5 (TGR5), with EC50s of 0.72 and 6.2 nM for hTGR5 and mTGR5, respectively. TC-G 1005 can reduce glucose levels in vivo[1][2].
Molecular Weight:
399.48
Purity:
99.83
CAS Number:
[1415407-60-1]
Formula:
C25H25N3O2
Target:
G protein-coupled Bile Acid Receptor 1
Application Notes:
Reference compound
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