LDN-209929 dihydrochloride is a potent and selective haspin kinase inhibitor (IC50=55 nM) with180-fold selectivity verses DYRK2 (IC50=9.9 µM). LDN-209929 is a optimized analogue of LDN-192960 (HY-13455)[2].
Molecular Weight:
405.77
Purity:
99
CAS Number:
[1784281-97-5]
Formula:
C17H19Cl3N2OS
Target:
DYRK,Haspin Kinase
Application Notes:
Reference compound
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