MS417 is a selective BET-specific BRD4 inhibitor, binds to BRD4-BD1 and BRD4-BD2 with IC50s of 30, 46 nM and Kds of 36.1, 25.4 nM, respectively, with weak selectivity at CBP BRD (IC50, 32.7 µM).
Molecular Weight:
414.91
Purity:
99.87
CAS Number:
[916489-36-6]
Formula:
C20H19ClN4O2S
Target:
Epigenetic Reader Domain,HIV
Application Notes:
Reference compound
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