EHT 5372 is a highly potent and selective inhibitor of DYRKs family kinases with IC50s of 0.22, 0.28, 10.8, 93.2, 22.8, 88.8, 59.0, 7.44, and 221 nM for DYRK1A, DYRK1B, DYRK2, DYRK3, CLK1, CLK2, CLK4, GSK-3alpha, and GSK-3beta, respectively[1][2].
Molecular Weight:
404.27
Purity:
98.12
CAS Number:
[1425945-63-6]
Formula:
C17H11Cl2N5OS
Target:
CDK,DYRK,GSK-3
Application Notes:
Reference compound
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