PLX51107 is a potent and selective BET inhibitor, with Kds of 1.6, 2.1, 1.7, and 5 nM for BD1 and 5.9, 6.2, 6.1, and 120 nM for BD2 of BRD2, BRD3, BRD4, and BRDT, respectively, PLX51107 also interacts with the bromodomains of CBP and EP300 (Kd, in the 10
Molecular Weight:
438.48
Purity:
99.74
CAS Number:
[1627929-55-8]
Formula:
C26H22N4O3
Target:
Epigenetic Reader Domain
Application Notes:
Reference compound
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