TP0463518 is a potent hypoxia-inducible factor prolyl hydroxylases (PHDs) inhibitor with a Ki value of 5.3 nM for human PHD2. TP0463518 also inhibits human PHD1/PHD3 with IC50s of 18 and 63 nM as well as monkey PHD2 with an IC50 value of 22 nM[1].
Molecular Weight:
431.83
Purity:
98.62
CAS Number:
[1558021-37-6]
Formula:
C20H18ClN3O6
Target:
HIF/HIF Prolyl-Hydroxylase
Application Notes:
Reference compound
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