IDH1 Inhibitor 1 is a potent, orally bioavailable, brain-penetrant and selective mutant IDH1 inhibitor with IC50s of 0.021 µM, 0.045 µM, and 2.52 µM for IDH1R132H, IDH1R132C, and IDH1WT, respectively[1]. Anticancer activity[1].
Molecular Weight:
450.39
Purity:
99.96
CAS Number:
[2234285-81-3]
Formula:
C20H18F4N6O2
Target:
Isocitrate Dehydrogenase (IDH)
Application Notes:
Reference compound
* VAT and and shipping costs not included. Errors and price changes excepted
