EN219 is a moderately selective synthetic covalent ligand against an N-terminal cysteine (C8) of RNF114 with an IC50 of 470 nM. EN219 inhibits RNF114-mediated autoubiquitination and p21 ubiquitination[1].
Molecular Weight:
456.56
Purity:
98.56
CAS Number:
[380351-29-1]
Formula:
C17H13Br2ClN2O
Target:
E1/E2/E3 Enzyme
Application Notes:
Reference compound
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