1G244 is a potent DPP8/9 inhibitor with IC50s of 12 nM and 84 nM, respectively. 1G244 does not inhibit DPPIV and DPPII. 1G244 induces apoptosis in multiple myeloma cells and has anti-myeloma effects[1][2].
Molecular Weight:
504.57
Purity:
98.66
CAS Number:
[847928-32-9]
Formula:
C29H30F2N4O2
Target:
Apoptosis,Dipeptidyl Peptidase
Application Notes:
Reference compound
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