GSK467 is a cell penetrant and selective KDM5B (JARID1B or PLU1) inhibitor with a Ki of 10 nM and an IC50 of 26 nM. GSK467 shows 180-fold selectivity for KDM4C and no measurable inhibitory effects toward KDM6 or other Jumonji family members[1][2].
Molecular Weight:
319.32
Purity:
98.14
CAS Number:
[1628332-52-4]
Formula:
C17H13N5O2
Target:
Histone Demethylase
Application Notes:
Reference compound
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