Thioperamide (MR-12842) is a potent, orally available, brain penetrant and selective H3 receptor antagonist with a Ki of 4.3 nM for inhibition of [3H]histamine release. Thioperamide inhibits [3H]histamine synthesis with a Ki of 31 nM[1].
Molecular Weight:
292.44
Purity:
99.91
CAS Number:
[106243-16-7]
Formula:
C15H24N4S
Target:
Histamine Receptor
Application Notes:
Reference compound
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