PCS1055 is a selective and competitive antagonist for muscarinic M4 receptor with an IC50 of 18.1 nM and a Kd of 5.72 nM. PCS1055 inhibits radioligand [3H]-NMS binding to the M4 receptor with a Ki of 6.5 nM. PCS1055 is also an inhibitor for AChE with IC5
Molecular Weight:
412.57
Purity:
98.02
CAS Number:
[357173-55-8]
Formula:
C27H32N4
Target:
Cholinesterase (ChE),mAChR
Application Notes:
Reference compound
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