AZ6102 is a potent dual TNKS1 and TNKS2 inhibitor, with IC50s of 3 nM and 1 nM, respectively, and alao has 100-fold selectivity against other PARP family enzymes, with IC50s of 2.0 µM, 0.5 µM, and >3 µM, for PARP1, PARP2, and PARP6, respectively.
Molecular Weight:
428.53
Purity:
99.65
CAS Number:
[1645286-75-4]
Formula:
C25H28N6O
Target:
PARP
Application Notes:
Reference compound
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