GNE-987, CAS [[2417371-71-0]]

Product Overview

• Article Name: GNE-987, CAS [[2417371-71-0]]
• Biozol Catalog Number: MCE-HY-129937A
• Supplier Catalog Number: HY-129937A
• Alternative Catalog Number: MCE-HY-129937A-10MG,MCE-HY-129937A-1MG,MCE-HY-129937A-5MG
• Manufacturer: MedchemExpress
• Category: Biochemikalien

Product Description

GNE-987 is a PROTAC connected by ligands for von Hippel-Lindau and BRD4. GNE-987 exhibits picomolar cell BRD4 degradation activity (DC50=0.03 nM for EOL-1 AML cell line). GNE-987 binds equipotently to the BD1 and BD2 bromodomains of BRD4 with low nanomol

Product Properties

• Molecular Weight: 1096.31
• Purity: 99.91
• CAS Number: [2417371-71-0]
• Formula: C56H67F2N9O8S2
• Target: Epigenetic Reader Domain,PROTACs

Application Notes

• Application Notes: Reference compound