Enpatoran (M5049) is a potent, orally active and dual TLR7/8 inhibitor with IC50s of 11.1 nM and 24.1 nM in HEK293 cells, respectively. Enpatoran is inactive against TLR3, TLR4 and TLR9. Enpatoran can block molecule synthetic ligands and natural endogeno
Molecular Weight:
320.31
Purity:
99.77
CAS Number:
[2101938-42-3]
Formula:
C16H15F3N4
Target:
Toll-like Receptor (TLR)
Application Notes:
Reference compound
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