TLK117, the active metabolite of TLK199, selective inhibits Glutathione S-transferase P1-1 (GSTP1-1) with a Ki of 0.4 µM for GSTP. TLK117 also competitively inhibits glyoxalase I with a Ki of 0.56 µM.
Molecular Weight:
473.54
Purity:
99.89
CAS Number:
[152684-53-2]
Formula:
C23H27N3O6S
Target:
Glutathione S-transferase
Application Notes:
Peptides
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