GSK046, CAS [[2474876-09-8]]

Product Overview

• Article Name: GSK046, CAS [[2474876-09-8]]
• Biozol Catalog Number: MCE-HY-136571
• Supplier Catalog Number: HY-136571
• Alternative Catalog Number: MCE-HY-136571-10MMX1ML,MCE-HY-136571-50MG,MCE-HY-136571-10MG,MCE-HY-136571-100MG,MCE-HY-136571-5MG,MCE-HY-136571-1MG,MCE-HY-136571-25MG
• Manufacturer: MedchemExpress
• Category: Biochemikalien
• Alternative Names: iBET-BD2

Product Description

GSK046 (iBET-BD2) is a potent, selective and orally active BD2 bromodomain inhibitor of the BET proteins, with IC50s of 264 nM (BRD2 BD2), 98 nM (BRD3 BD2), 49 nM (BRD4 BD2) and 214 nM (BRDT BD2), respectively. GSK046 has immunomodulatory activity[1].

Product Properties

• Molecular Weight: 414.47
• Purity: 99.65
• CAS Number: [2474876-09-8]
• Formula: C23H27FN2O4
• Target: Epigenetic Reader Domain

Application Notes

• Application Notes: Reference compound