RP101075, an active metabolite of Ozanimod, is a potent, orally active S1PR (sphingosine-1-phosphate receptor 1) agonist, with an EC50 of 0.27 nM. RP101075 displays >100-fold selectivity over S1PR5 (EC50=5.9 nM) and >10000-fold over S1PR 2, 3, and 4. RP1
Molecular Weight:
360.41
CAS Number:
[1306760-73-5]
Formula:
C21H20N4O2
Target:
Drug Metabolite,LPL Receptor
Application Notes:
Reference compound
* VAT and and shipping costs not included. Errors and price changes excepted