NBI-42902 is an orally active, potent functional and competitive antagonist of GnRH receptor with an IC50 value of 0.79 nM, a Ki value of 0.56 nM, respectively. NBI-42902 inhibits GnRH-stimulated inositol phosphate (IP) accumulation, Ca2+ flux, and ERK1/
Molecular Weight:
495.49
Purity:
98.65
CAS Number:
[352290-60-9]
Formula:
C27H24F3N3O3
Target:
GnRH Receptor,PERK
Application Notes:
Reference compound
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