Aldumastat (GLPG1972, S201086) is a potent, seletive and orally active ADAMTS-5 (IC50=19 nM) inhibitor, and has 8-fold seletivity over ADAMTS-4 (IC50=156 nM). Aldumastat has anticatabolic activity and is used for osteoarthritis research[1].
Molecular Weight:
406.43
Purity:
99.54
CAS Number:
[1957278-93-1]
Formula:
C20H24F2N4O3
Target:
ADAMTS
Application Notes:
Reference compound
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