GSK973 is a highly selective, orally bioavailable inhibitor of the BD2s (second bromodomains) of the BET family, with a pIC50 of 7.8 and a pKd of 8.7 for BRD4 BD2. GSK973 displays a 1600-fold selectivity for BRD4 BD2 over BRD4 BD1. GSK973 shows good pote
Molecular Weight:
410.44
Purity:
99.46
CAS Number:
[2138473-38-6]
Formula:
C23H23FN2O4
Target:
Epigenetic Reader Domain
Application Notes:
Reference compound
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