MRTX-1719 is a potent, orally active, selective PRMT5MTA complex inhibitor, with IC50 of 3.6 and 20.5 nM for PRMT5MTA and PRMT5. MRTX-1719 binds to the PRMT5MTA complex, with KD value of 0.14 pM. MRTX-1719 shows antineoplastic activity in vitro and in
Molecular Weight:
464.88
Purity:
99.40
CAS Number:
[2630904-45-7]
Formula:
C23H18ClFN6O2
Target:
Histone Methyltransferase
Application Notes:
Reference compound
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