CCG258747 is a selective GRK2 inhibitor (IC50=18 nM) with high selectivity over GRK1, GRK5, PKA, and ROCK1 (518, 83, >5500, and >550-fold, respectively).CCG258747 also blocks the internalization of the µ-opioid receptor. G protein-coupled receptor (GPCR)
Molecular Weight:
502.54
Purity:
99.17
CAS Number:
[2615910-00-2]
Formula:
C28H27FN4O4
Target:
Opioid Receptor
Application Notes:
Reference compound
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