I-BET567 is a potent and orally active inhibitor of pan-BET candidate with pIC50s of 6.9 and 7.2 for BRD4 BD1 and BD2, respectively. I-BET567 has been demonstrated efficacy in mouse models of oncology and inflammation[1].
Molecular Weight:
359.81
Purity:
99.49
CAS Number:
[1887237-54-8]
Formula:
C17H18ClN5O2
Target:
Epigenetic Reader Domain
Application Notes:
Reference compound
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