LX-039 is a highly potent, selective and orally active estrogen receptor degrader with EC50 value of 2.29 nM. LX-039 has indole C-3 chlorine atom. LX-039 exhibits excellent mouse pharmacokinetics, low clearance, high Cmax and oral exposure. LX-039 has an
Molecular Weight:
480.36
CAS Number:
[2135341-09-0]
Formula:
C27H20Cl2FNO2
Target:
Estrogen Receptor/ERR
Application Notes:
Reference compound
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