CDK8-IN-12 is an orally active, potent CDK8 inhibitor with a Ki of 14 nM. CDK8-IN-12 has off-target kinase inhibition on GSK-3alpha, GSK-3beta, PCK-theta with Kis of 13 nM, 4 nM, 109 nM, respectively. CDK8-IN-12 shows potent anti-proliferative effects selectively o
Molecular Weight:
381.86
Purity:
99.74
CAS Number:
[2613307-67-6]
Formula:
C21H20ClN3O2
Target:
CDK,GSK-3,PKC
Application Notes:
Reference compound
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