Dim16 is a dual PCSK9/HMG-CoAR inhibitor, with an IC50 value of 19 nM for PCSK9. Dim16 inhibits PCSK9-LDLR binding with an IC50 value of 0.8 nM. Dim16 increases LDL uptake in HepG2 cells[1].
Molecular Weight:
583.55
CAS Number:
[2743448-32-8]
Formula:
C29H38IN5
Target:
Ser/Thr Protease
Application Notes:
Reference compound
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