Smurf1-IN-1 is an orally active and selective inhibitor of specific E3 ubiquitin protein ligase 1 (SMURF1) with an IC50 of 92 nM. Smurf1-IN-1 has significant efficacy in rats model of pulmonary hypertension[1].
Molecular Weight:
468.98
Purity:
99.47
CAS Number:
[1824708-03-3]
Formula:
C24H29ClN6O2
Target:
E1/E2/E3 Enzyme
Application Notes:
Reference compound
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