D3R/MOR antagonist 1 (Compound 114) is a D3R/MOR antagonist (Ki: 46.5 nM and 691 nM respectively). D3R/MOR antagonist 1 has the potential to produce analgesic effects through MOR partial agonism, reduce opioid-misuse liability via D3R antagonism[1].
Molecular Weight:
420.38
Formula:
C22H27Cl2N3O
Target:
Dopamine Receptor,Opioid Receptor
Application Notes:
Reference compound
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