CVN417 is an orally active alpha6 subunit-containing nAChR antagonist, modulating phasic dopaminergic neurotransmission in an impulse-dependent manner. CVN417 inhibits Ca(2+) effluents mediated by nAChR subunits with IC50s of 0.086 µM (alpha6), 2.56 µM (alpha3) and
Molecular Weight:
362.85
CAS Number:
[2919851-73-1]
Formula:
C18H23ClN4O2
Target:
nAChR
Application Notes:
Reference compound
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