PBRM1-BD2-IN-5 is a potent PBRM1 Bromodomain inhibitor with Kd values of 1.5 µM and 3.9 µM for PBRM1-BD2 and PBRM1-BD5, respectively, and an IC50 value of 0.26 µM for PBRM1-BD2. PBRM1-BD2-IN-5 reduces the binding of full-length PBRM1 within the PBAF comp
Molecular Weight:
272.73
Purity:
99.55
CAS Number:
[2819989-61-0]
Formula:
C15H13ClN2O
Target:
Epigenetic Reader Domain
Application Notes:
Reference compound
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