PHD-IN-1 (compound 80) is a potent inhibitor of PHD2,with an IC50 value of 5 nM. PHD-IN-1 shows EC50s of 2.5 µM in EPO Elisa assay both in Caco2-HIFla-HiBiT-clone-1 cells and Hep3B cells,respectively[1].
Molecular Weight:
441.49
CAS Number:
[2924182-31-8]
Formula:
C24H23N7O2
Target:
HIF/HIF Prolyl-Hydroxylase
Application Notes:
Reference compound
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