CH5164840 (16) shows high binding affinity for N-terminal Hsp90a (Kd = 0.52 nM) and strong anti-proliferative activity against human cancer cell lines (HCT116 IC50 = 0.15 µM, NCI-N87 IC50 = 0.066 µM). CH5164840 (16) is orally active (t1/2 = 2.64 h) with
Molecular Weight:
385.48
CAS Number:
[1052645-73-4]
Formula:
C19H23N5O2S
Target:
HSP
Application Notes:
Reference compound
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