Dagrocorat (PF-00251802) is an orally active and selective high-affinity partial agonist of the glucocorticoid receptor. Dagrocorat is also a time-dependent reversible inhibitor of CYP3A (IC50=1.3 µM in human liver microsomes) and CYP2D6 (Ki=0.57 µM in h
Molecular Weight:
494.55
Purity:
99.90
CAS Number:
[1044535-52-5]
Formula:
C29H29F3N2O2
Target:
Cytochrome P450,Glucocorticoid Receptor
Application Notes:
Reference compound
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