Grapiprant (CJ-023423) is a selective EP4 receptor antagonist whose physiological ligand is prostaglandin E2 (PGE2). Grapiprant displaces [3H]-PGE2 (1 nM) binding to dog recombinant EP4 receptor with IC50 value of 35 nM and Ki value of 24 nM. Grapiprant
Molecular Weight:
491.61
Purity:
99.57
CAS Number:
[415903-37-6]
Formula:
C26H29N5O3S
Target:
Prostaglandin Receptor
Application Notes:
Reference compound
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