GSK180736A is potent Rho-associated coiled-coil kinase 1 (ROCK1) inhibitor with an IC50 of 100 nM. GSK180736A is also a selective and ATP-competitive G protein-coupled receptor kinase 2 (GRK2) inhibitor with an IC50 of 0.77 µM.
Molecular Weight:
365.36
Purity:
98.01
CAS Number:
[817194-38-0]
Formula:
C19H16FN5O2
Target:
ROCK
Application Notes:
Reference compound
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