JKC363, a selective melanocortin MC4 receptor antagonist, has a 90-fold higher affinity at the MC4 receptor (IC50=0.5 nM) than at the MC3 receptor (44.9 nM). JKC-363 blocks the stimulatory effect of alpha-MSH on TRH release. Anti-hyperalgesic effect[1][2].
Molecular Weight:
1506.71
Purity:
99.55
CAS Number:
[436083-30-6]
Formula:
C69H91N19O16S2
Target:
Melanocortin Receptor
Application Notes:
Peptides
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