Targefrin is a potent EphA2-targeting agent, acts as an antagonist. Targefrin binds EphA2-LBD with 21 nM dissociation constant and an IC50 value of 10.8 nM. Targefrin induces cellular receptor internalization and degradation in several pancreatic cancer
Molecular Weight:
1700.94
Purity:
99.45
CAS Number:
[3031514-44-7]
Formula:
C85H116F3N19O15
Target:
Ephrin Receptor
Application Notes:
Peptides
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