GI-530159 is a selective opener of TREK1 and TREK2 potassium channels. GI-530159 displays selectivity for TREK1/2 over TRAAK, TASK3 and other potassium channels, with an EC50 of 0.76 µM for TREK1. GI-530159 reduces rat dorsal root ganglion neuron excitab
Molecular Weight:
518.45
Purity:
99.27
CAS Number:
[69563-88-8]
Formula:
C27H20F6N2O2
Target:
Potassium Channel
Application Notes:
Reference compound
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