YKL-5-124

Catalog Number: SEL-S8863
Article Name: YKL-5-124
Biozol Catalog Number: SEL-S8863
Supplier Catalog Number: S8863
Alternative Catalog Number: SEL-S8863-10MM/1ML,SEL-S8863-25MG,SEL-S8863-5MG
Manufacturer: Selleck
Category: Biochemikalien
YKL-5-124 is a potent, selective and covalent CDK7 inhibitor with an IC50 of 9.7 nM, 1300 nM and 3020 nM for inhibiting CDK7/Mat1/CycH, CDK2 and CDK9 respectively. It displays biochemical and cellular selectivity for CDK7 over CDK12/13.
CAS Number: [1957203-01-8]