Aprocitentan D4 (ACT-132577 D4) is a deuterium-labeled Aprocitentan. Aprocitentan is a major and pharmacologically active metabolite of Macitentan. Aprocitentan is a dual ETA/ETB antagonist (IC50s: 3.4 nM and 987 nM, pA2s: 6.7 and 5.5).
Molecular Weight:
550.22
CAS Number:
[T10351]
Formula:
C16H10D4Br2N6O4S
Target:
ACT-132577 D4
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