AR-A 2 is a selective 5-HT1B receptor antagonist, with a high affinity to guinea pig cortex 5HT1B/1D and recombinant guinea pig 5-HT1B receptors (Ki: 0.24 and 0.47 nM) and with 10-fold lower affinity to guinea pig 5-HT1D receptor (Ki: 5 nM).
Molecular Weight:
448.6
CAS Number:
[220051-79-6]
Formula:
C27H36N4O2
Target:
AR-A 000002
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