LT052, a highly active and selective BET BD1 inhibitor with an IC50 of 87.7 nM, demonstrates nanomolar BRD4 BD1 potency and significant selectivity, being 138-fold more selective for BRD4 BD1 over BRD4 BD2 (IC50 =12.130 µM). Its anti-inflammatory propert
Molecular Weight:
449.48
CAS Number:
[2543545-44-2]
Formula:
C22H19N5O4S
Target:
Epigenetic Reader Domain
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