Talmapimod (SCIO-469) is an selective, orally active, and ATP-competitive p38alpha inhibitor with IC50 of 9 nM and 90 nM for p38alpha and p38beta, respectively. Talmapimod exhibits at least 2000-fold selectivity over a panel of 20 kinases, including other MAPKs.
Molecular Weight:
513
CAS Number:
[309913-83-5]
Formula:
C27H30ClFN4O3
Target:
p38 MAPK
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