Sitravatinib malate, CAS [[2244864-88-6]]
Catalog Number:
TGM-T12925
Article Name: |
Sitravatinib malate, CAS [[2244864-88-6]] |
Biozol Catalog Number: |
TGM-T12925 |
Supplier Catalog Number: |
T12925 |
Alternative Catalog Number: |
TGM-T12925-25MG,TGM-T12925-50MG,TGM-T12925-100MG |
Manufacturer: |
TargetMol |
Category: |
Biochemikalien |
Alternative Names: |
MGCD516 malate |
Sitravatinib malate is an orally bioavailable receptor inhibitor of tyrosine kinase (RTK) (IC50s of 1.5 nM, 2 nM, 2 nM, 5 nM, 6 nM, 6 nM, 8 nM, 0.5 nM, 29 nM, 5 nM, and 9 nM for Axl, MER, VEGFR3, VEGFR2, VEGFR1, KIT, FLT3, DDR2, DDR1, TRKA, TRKB, respect |
Molecular Weight: |
763.76 |
CAS Number: |
[2244864-88-6] |
Formula: |
C37H35F2N5O9S |
Target: |
TAM Receptor |