Darigabat (PF-06372865) is an orally active and selective GABAA receptor modulator that crosses the blood-brain barrier and exhibits anxiolytic activity, with Ki values of 2.9 nM, 21 nM, and 134 nM for alpha2, alpha1 PAM, and alpha2 PAM, respectively.Darigabat is us
Molecular Weight:
440.49
CAS Number:
[1614245-70-3]
Formula:
C22H21FN4O3S
Target:
CVL-865 , PF-6372865 , PF-06372865
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